Suggestions

Du même auteur

Biologically active carbazole derivatives: focus on oxazinocarbazoles and related compounds

Archive ouverte | Bouaziz, Zouhair | CCSD

International audience

Uncompetitive nanomolar dimeric indenoindole inhibitors of the human breast cancer resistance pump ABCG2

Archive ouverte | Guragossian, Nathalie | CCSD

International audience. Multidrug resistance membrane pumps reduce the efficacy of chemotherapies by exporting a wide panel of structurally-divergent drugs. Here, to take advantage of the polyspecificity of the huma...

Converting potent indeno[1,2-b]indole inhibitors of protein kinase CK2 into selective inhibitors of the breast cancer resistance protein ABCG2

Archive ouverte | Jabor Gozzi, Gustavo | CCSD

International audience. A series of indeno[1,2-b]indole-9,10-dione derivatives were synthesized as human casein kinase II (CK2) inhibitors. The most potent inhibitors contained a N(5)-isopropyl substituent on the C-...

Chargement des enrichissements...