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Archive ouverte | Jabor Gozzi, Gustavo | CCSD

International audience. A series of indeno[1,2-b]indole-9,10-dione derivatives were synthesized as human casein kinase II (CK2) inhibitors. The most potent inhibitors contained a N(5)-isopropyl substituent on the C-...

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Archive ouverte | Gozzi, Gustavo Jabor | CCSD

International audience. Ketonic indeno[1,2-b]indole-9,10-dione derivatives, initially designed as human casein kinase II (CK2) inhibitors, were recently shown to be converted into efficient inhibitors of drug efflux...

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Archive ouverte | Bouaziz, Zouhair | CCSD

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